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Department of Pharmacy

Guru Ghasidas Vishwavidyalaya, Bilaspur | School of Studies of Natural Resources

Dr. Sanjay Kumar Bharti

  • Associate Professor
  • sanjay.itbhu@gmail.com
  • 9301808566

Personal Information

  • Full Name: Dr. Sanjay Kumar Bharti
  • Mobile Number: 9301808566
  • EmailID: sanjay.itbhu@gmail.com
  • Designation: Associate Professor
Qualification

  • 2011
    Ph. D.

    IIT(BHU)-Varanasi

  • 2006
    M. Pharm.

    RGPV, Bhopal

  • 2003
    B. Pharm.

    IIT(BHU)-Varanasi

Experience

  • 2024 - 2025
    Associate Professor

    Guru Ghasidas Vishwavidyalaya (A Central University)

  • 2012 - 2024
    Assistant Professor

    Guru Ghasidas Vishwavidyalaya (A Central University)

  • 2010 - 2012
    Lecturer

    National Institute of Pharmaceutical Education and Research (NIPER), Hajipur

Doctoral Theses Guided

Design, synthesis and biological evaluation of newer thiazolidine-2,4-diones as anticancer agents

  • Guru Ghasidas Vishwavidyalaya (A Central University)

  • Mr. Vivek Asati

Research Projects

Design and synthesis of some novel metal (Co, Ni, Ga) complexes of bi-/tridentate ligand(s) as potential nucleolytic and anticancer agents

Completed Amount: ₹6.00

Funding Agency: UGC, New Delhi

Duration : 01:04:2013 - 31:03:2015

Publications

An updated patent review on rational combinations of HDAC inhibitors for cancer chemotherapy (2020 – present): part 1-patent granted

Yugal Kishor Shukla, Vandana, Vivekananda Mandal, Vivek Asati, Raj K. Keservani, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Expert Opinion on Therapeutic Patents

Year: 2025

DOI: https://doi.org/10.1080/13543776.2025.2546595

Impact Factor: 5.40

An updated patent review on rational combinations of HDAC inhibitors for cancer chemotherapy (2020 – present): part 2 - patent published

Yugal Kishor Shukla, Vandana, Vivekananda Mandal, Vivek Asati, Raj K. Keservani, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Expert Opinion on Therapeutic Patents

Volume: 35(8)

Year: 2025

Pages: 875–900

Impact Factor: 5.40

Structural aspects of HIV-1 integrase inhibitors: SAR studies and synthetic strategies

Barik, Pallavi, Shankar Gupta, Gurpreet Singh, Sanjay Kumar Bharti, and Vivek Asati

Publication Type: Journal Article (International)

Journal: Molecular Diversity

Volume: 29

Year: 2025

Pages: 4963–4997

DOI: https://doi.org/10.1007/s11030-024-11068-4

Link

Impact Factor: 3.80

MEK Inhibitors in Oncology: A Patent Review and Update (2016 – Present)

Anjali Suryavanshi, Vandana, Yugal Kishor Shukla, Vipul Kumar, Pragya Gupta, Vivek Asati, Debarshi Kar Mahapatra, Raj K. Keservani, Sanmati Kumar Jain, and Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Expert Opinion on Therapeutic Patents

Volume: 34

Year: 2024

Pages: 963–1007

DOI: https://doi.org/10.1080/13543776.2024.2403634

Link

Impact Factor: 4.60

PIM Kinase Inhibitors: An Updated Patent Review (2016-Present)

Anushka Sharma, Rahul Dubey, Shankar Gupta, Vivek Asati, Vipul Kumar, Dileep Kumar, Debarshi Kar Mahapatra, Meenakshi Jaiswal, Sanmati Kumar Jain, and Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: . Expert Opinion on Therapeutic Patents

Volume: 34

Year: 2024

Pages: 365–82

DOI: doi: 10.1080/13543776.2024.2365411

Link

Impact Factor: 4.60

Recent Advances in the Treatment and Management of Alzheimer’s Disease: A Precision Medicine Perspective

Deepali Shukla, Anjali Suryavanshi, Sanjay Kumar Bharti*, Vivek Asati and Debarshi Kar Mahapatra

Publication Type: Journal Article (International)

Journal: Current Topics in Medicinal Chemistry

Volume: 24

Year: 2024

Pages: 1699-1737

DOI: doi: 10.2174/0115680266299847240328045737

Link

Impact Factor: 2.90

3D-QSAR and Pharmacophoric study on 2,6-Disubstituted Thiazolo [4,5-b] Pyridines as H3 Receptor Antagonists

S. K. Jain, S. K. Bharti, B.G.V.S. Jagan, Ajay K. Gupta

Publication Type: Journal Article (International)

Journal: Research Journal of Pharmacy and Technology (RJPT),

Volume: 16

Year: 2023

Pages: 4575-4582

DOI: 10.52711/0974-360X.2023.00745

Link

Recent advances of PI3 Kinase inhibitors: Structure anticancer activity relationship studies

Asati Vivek, Anant Arjun, Mahapatra Kar Debarshi and Bharti Kumar Sanjay

Publication Type: Journal Article (International)

Journal: Mini-Reviews in Medicinal Chemistry

Volume: 22

Year: 2022

Pages: 2146 - 2165

DOI: doi: 10.2174/1389450123666220202154757.

Link

Impact Factor: 3.80

Discovery of novel ALK2 inhibitors of pyrazolo-pyrimidines: A computational study

Vivek Asati, Sanjay K. Bharti, Ratnesh Das, Varsha Kashaw & Sushil Kumar Kashaw

Publication Type: Journal Article (International)

Journal: Journal of Biomolecular Structure and Dynamics

Volume: 40

Year: 2022

Pages: 10422-10436

DOI: 10.1080/07391102.2021.1944320

Link

Impact Factor: 5.30

Recent progress in theranostic nanoparticles for personalized medicine,

Krishna Kant Jangde, Anjali Suryavanshi, Deepali Shukla, Meenakshi Jaiswal, Vipul Kumar, Sanjay Kumar Bharti

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 19

Year: 2022

Pharmacovigilance in digital era: real-world data and safety monitoring

Vipul Kumar, Sanjay Kumar Bharti*, Deepali Shukla, Anjali Suryavanshi, Krishna Kant Jangde, Karthikeyan Kesavan, Vivek Asati, Debarshi Kar Mahapatra , Raj K. Keservani

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 28

Year: 2021

Pages: 1197–1202

DOI: 10.1002/cpt.2172

Link

Synthesis, Characterized and Biological Evaluation of Some Novel Schiff Bases,

None

Publication Type: Journal Article (International)

Journal: International Research Journal of Engineering and Technology (IRJET),

Volume: 8

Year: 2021

Pages: 931-939

Link

Current discovery progress of some emerging anti-infective chalcones

13. Debarshi Kar Mahapatra, Soumajit Ghorai, Sanjay Kumar Bharti, Asmita Gajbhiye Patil and Shovanlal Gayen,

Publication Type: Journal Article (International)

Journal: Current Drug Discovery Technologies

Volume: 17

Year: 2020

Pages: 30-44

DOI: 10.2174/1570163815666180720170030

Link

An updated patent review of therapeutic applications of chalcone derivatives (2014-present),

Debarshi Kar Mahapatra, Vivek Asati, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Expert Opinion on Therapeutic Patents

Volume: 29

Year: 2019

Pages: 385-406

DOI: 10.1080/13543776.2019.1613374

Link

Impact Factor: 6.60

Perspectives of medicinally privileged chalcone based metal coordination compounds for biomedical applications

Debarshi Kar Mahapatra, Sanjay Kumar Bharti*, Vivek Asati, Sushil Kumar Singh

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 174

Year: 2019

Pages: 142-158

DOI: https://doi.org/10.1016/j.ejmech.2019.04.032

Link

Impact Factor: 7.00

PIM Kinase Inhibitors: Structural and Pharmacological Perspectives.

Vivek Asati, Debarshi Kar Mahapatra, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 15

Year: 2019

Pages: 172:95-108

DOI: doi: 10.1016/j.ejmech.2019.03.050.

Link

Impact Factor: 7.00

3D-QSAR and molecular docking studies on oxadiazole substituted benzimidazole derivatives: Validation of experimental inhibitory potencies towards COX-2,

Vivek Asati, Piyush Ghode, Shalini Bajaj, Sanmati Kumar Jain, Sanjay Kumar Bharti*,

Publication Type: Journal Article (International)

Volume: 15

Year: 2019

Pages: 277-293

DOI: doi: 10.2174/1573409914666181003153249.

Link

Impact Factor: 1.60

Recent therapeutic progress of chalcone scaffold bearing compounds as prospective anti-gout candidates

Debarshi Kar Mahapatra, Vivek Asati, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Journal of Critical Reviews

Volume: 6

Year: 2019

Pages: 1-5

DOI: 10.22159/jcr.2019v6i1.31760

Link

Impact Factor: 1.40

Nutritional advantages and effects of vitamins in human health

Khemchand R. Surana , Eknath D. Ahire, Raj K. Keservani, Arvind Kumar Gupta, Meenendra Tripathi, Akanksha Yadav, Sanjay K. Bharti5*, Brijesh Kumar Singh, Nagendra Shukla

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 16

Year: 2019

Pages: 67-70

Virtual Screening, Molecular Docking, and DFT Studies of Some Thiazolidine-2,4-diones as Potential PIM-1 Kinase Inhibitors,

None

Publication Type: Journal Article (International)

Journal: ChemistrySelect

Volume: 3

Year: 2018

Pages: 12186-12194

DOI: https://doi.org/10.1002/slct.201702392

Link

Impact Factor: 2.30

Design, synthesis and molecular modeling studies of novel thiazolidine-2,4-dione derivatives as potential anti-cancer agents

Vivek Asati, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Journal of Molecular Structure

Volume: 1154

Year: 2018

Pages: 406-417

DOI: https://doi.org/10.1016/j.molstruc.2017.10.077

Link

Impact Factor: 3.80

Overview on gastro retentive drug delivery systems: Current scenario and future prospective

Rashmi Chourasiya, Meenakshi Jaiswal, Sanjay Kumar Bharti , Sanmati Kumar Jain , Ajay Kumar Gupta , Nidhi Agrawal

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 15

Year: 2018

Pages: 132-135

Microwave in synthetic chemistry: a green chemistry approach,

Sanjay Kumar Bharti1* , Meenakshi Jaiswal , N.S. Hari Narayana Moorthy

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 15

Year: 2018

Pages: 124-131

Design, microwave assisted synthesis and characterization of benzimidazolin-2-one and its derivatives,

Sanjay Kumar Bharti1* , Meenakshi Jaiswal , N.S. Hari Narayana Moorthy

Publication Type: Journal Article (National)

Journal: Chhattisgarh Journal of Science and Technology

Volume: 15

Year: 2018

Pages: 92-96

MEK inhibitors in oncology: a patent review (2015-Present),

Debarshi Kar Mahapatra, Vivek Asati and Sanjay Kumar Bharti*

Publication Type: Journal Article (International)

Journal: Expert Opinion on Therapeutic Patents

Volume: 27

Year: 2017

Pages: 887-906

DOI: 10.1080/13543776.2017.1339688.

Link

Impact Factor: 6.60

Chalcone derivatives: anti-inflammatory potential and molecular targets perspectives

Debarshi Kar Mahapatra, Sanjay Kumar Bharti* and Vivek Asati

Publication Type: Journal Article (International)

Journal: Current Topics in Medicinal Chemistry

Volume: 17

Year: 2017

Pages: 3146-3169.

DOI: 10.2174/1568026617666170914160446.

Link

Impact Factor: 3.57

Nature inspired green fabrication technology for silver nanoparticles

Debarshi Kar Mahapatra*, Sanjay Kumar Bharti, Vivek Asati,

Publication Type: Journal Article (International)

Journal: Current Nanomedicine

Volume: 7

Year: 2017

Pages: 5-24

DOI: https://doi.org/10.2174/2468187306666160927122028

Link

K-Ras and its inhibitors towards personalized cancer treatment: Pharmacological and structural perspectives,

Vivek Asati, Debarshi Kar Mahapatra and Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 125

Year: 2017

Pages: 299-314

DOI: https://doi.org/10.1016/j.ejmech.2016.09.049

Link

Impact Factor: 7.00

3D-QSAR and virtual screening studies of thiazolidine-2,4-dione analogs: Validation of experimental inhibitory potencies towards PIM-1 kinase

Vivek Asati, Sanjay Kumar Bharti, Ashok Kumar Budhwani

Publication Type: Journal Article (International)

Journal: Journal of Molecular Structure

Volume: 11335

Year: 2017

Pages: 278-293

DOI: https://doi.org/10.1016/j.molstruc.2016.12.006

Link

Impact Factor: 3.84

SWFB and GA strategies for variable selection in QSAR studies for the validation of thiazolidine-2,4-dione derivatives as promising antitumor candidates

Vivek Asati, Sanjay Kumar Bharti, Ankita Rathore, Debarshi Kar Mahapatra

Publication Type: Journal Article (National)

Journal: Indian Journal of Pharmaceutical Education and Research

Volume: 51

Year: 2017

Pages: 436-451

DOI: doi:10.5530/ijper.51.3.72

Link

Impact Factor: 0.60

Novel Murrayanine based Pyrazole analogs as emerging anti-fungal candidates: Design, synthesis, characterization, and in vitro evaluation

Debarshi Kar Mahapatra, Ruchi S. Shivhare, Sanjay K. Bharti

Publication Type: Journal Article (International)

Journal: Research Pharmaceutica

Volume: 1

Year: 2017

Pages: 1-5

Molecular Modeling Studies of Some Thiazolidine-2, 4-dione Derivatives as 15-PGDH Inhibitors

Vivek Asati, Shalini Bajaj, Debarshi Kar Mahapatra, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Medicinal Chemistry Research

Volume: 25

Year: 2016

Pages: 94-108

DOI: https://doi.org/10.1007/s00044-015-1442-5

Link

Impact Factor: 2.50

PI3K/Akt/mTOR and Ras/Raf/MEK/ERK Signaling Pathways Inhibitors as Anticancer Agents: Structural and Pharmacological Perspectives

Vivek Asati, Debarshi Kar Mahapatra, Sanjay Kumar Bharti*,

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 109

Year: 2016

Pages: 314-341

DOI: https://doi.org/10.1016/j.ejmech.2016.01.012

Link

Impact Factor: 7.00

Therapeutic Potential of Chalcones as Cardiovascular Agents

Debarshi Kar Mahapatra, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Life Science

Volume: 148

Year: 2016

Pages: 154–172

DOI: https://doi.org/10.1016/j.lfs.2016.02.048

Link

Impact Factor: 6.70

QSAR studies for some thiazolidine-2,4-dione derivatives as PIM-2 kinase inhibitors

Vivek Asati*, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Medicinal Chemistry Research

Volume: 25

Year: 2016

Pages: 1329-1339

DOI: https://doi.org/10.1007/s00044-016-1577-z

Link

Impact Factor: 2.35

Mutant B-Raf Kinase inhibitors as anticancer agents

Vivek Asati*, Sanjay Kumar Bharti, Debarshi Kar Mahapatra

Publication Type: Journal Article (International)

Journal: Anti-cancer agents in medicinal chemistry

Volume: 16

Year: 2016

Pages: 1558-1575

DOI: 10.2174/1871520616666160606101848

Link

Impact Factor: 2.50

Triggering PIK3CA mutations in PI3K/AKT/mTOR axis: Exploration of newer inhibitors and rational preventive strategies

Vivek Asati, Sanjay Kumar Bharti, Debarshi Kar Mahapatra, Ashok Kumar Budhwani

Publication Type: Journal Article (International)

Journal: Current Pharmaceutical Design

Volume: 22

Year: 2016

Pages: 6039-6054

DOI: 10.2174/1381612822666160614000053

Link

Impact Factor: 3.30

Chalcone scaffolds as anti-infective agents: Structural and molecular target perspectives

Debarshi Kar Mahapatra, Sanjay Kumar Bharti*, Vivek Asati,

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 101

Year: 2015

Pages: 496-524

DOI: https://doi.org/10.1016/j.ejmech.2015.06.052

Link

Impact Factor: 7.00

Anti-cancer chalcones: Structural and molecular target perspectives

Debarshi Kar Mahapatra, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 98

Year: 2015

Pages: 69-114

DOI: https://doi.org/10.1016/j.ejmech.2015.05.004

Link

Impact Factor: 7.00

Chalcones and Their Therapeutic Targets for the Management of Diabetes: Structural and Pharmacological Perspectives

Debarshi Kar Mahapatra, Vivek Asati, Sanjay K. Bharti

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 92

Year: 2015

Pages: 839-865

DOI: https://doi.org/10.1016/j.ejmech.2015.01.051

Link

Impact Factor: 7.00

Mutations in surface protein of swine flu: A major problem for H1N1 inhibitor

Mukesh Kumar Gupta, J.S. Dangi, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Asian Journal of Biomedical and Pharmaceutical Sciences

Volume: 5

Year: 2015

Pages: 1-9

Thiazolidine-2,4-diones as multi-targeted scaffold in medicinal chemistry: Potential anticancer agents

Vivek Asati, Debarshi Kar Mahapatra, Sanjay K. Bharti

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 87

Year: 2014

Pages: 814 – 833

DOI: https://doi.org/10.1016/j.ejmech.2014.10.025

Link

Impact Factor: 7.00

Design, synthesis and biological evaluation of some novel benzylidene-2-(4-phenylthiazol-2-yl) hydrazines as potential anti-inflammatory agents,

Sanjay K. Bharti*, Sushil K. Singh

Publication Type: Journal Article (International)

Journal: Medicinal Chemistry Research

Volume: 23

Year: 2014

Pages: 1004-1015

DOI: https://doi.org/10.1007/s00044-013-0708-z

Link

Impact Factor: 2.30

Drug of choice for swine flu: a challenge ahead

Mukesh Kumar Gupta, Jawahar Singh Dangi, Sanjay Kumar Bharti, Krisna Gopal P

Publication Type: Journal Article (International)

Journal: Asian Journal of Pharmaceutical Sciences and Research

Volume: 3

Year: 2013

Pages: 01-18

Histamine H4 Receptor: A Novel Target for Inflammation Therapy

C. Saravanan, Sanjay Kumar Bharti, S. Jaggi, S. K. Singh

Publication Type: Journal Article (International)

Journal: Mini-Reviews in Medicinal Chemistry

Volume: 11

Year: 2011

Pages: 143 - 158

DOI: DOI: 10.2174/138955711794519519

Link

Impact Factor: 3.80

Pharmacogeomics in clinical research and practice: An ethical consideration

Ajay Verma*, Tanu Khurana, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Pharmacologyonline,

Volume: 1

Year: 2011

Pages: 453-461

Homology modeling and molecular dynamics study of serine hydroxyl methyl transferase enzyme from Leishmania donovani

Ashish Sethi, Rakesh Kumar Sharma, Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Journal of Pharmacy Research

Volume: 4

Year: 2011

Pages: 2269-2272

Synthesis, characterization, DNA cleavage and in vitro antimicrobial activities of novel copper(II) complexes of Schiff bases containing a 2,4-disubstituted thiazole

Sanjay Kumar Bharti, Saurabh K. Patel, Gopal Nath, Ragini Tilak, Sushil K. Singh*,

Publication Type: Journal Article (International)

Journal: Transition Metal Chemistry

Volume: 35

Year: 2010

Pages: 917 – 925

DOI: https://doi.org/10.1007/s11243-010-9412-8

Link

Impact Factor: 1.60

Synthesis, antibacterial and antifungal activities of some novel Schiff bases containing 2, 4-disubstituted thiazole ring

Sanjay Kumar Bharti, G. Nath, R. Tilak and S. K. Singh

Publication Type: Journal Article (International)

Journal: European Journal of Medicinal Chemistry

Volume: 45

Year: 2010

Pages: 651 – 660

DOI: https://doi.org/10.1016/j.ejmech.2009.11.008

Link

Impact Factor: 7.00

2D – Quantitative Structure Property Relationship (QSPR) Study of N-(aryl)-2-thiophen-2-ylacetamide Derivatives as Antitubercular Agents

Hemendra Singh Chouhan, Sanjay Kumar Bharti, Sushil K. Singh

Publication Type: Journal Article (International)

Journal: Asian Journal of Chemistry

Volume: 22

Year: 2010

Pages: 4675-4680

Synthesis and Evaluation of N-Mannich bases of Isatin-3- (4- aldehyde/ketone 2-thiosemicarbazones) derivatives as potent anticonvulsant agents

S. K. Singh, S. Jaggi, Sanjay Kumar Bharti and R. G. Kulkarni

Publication Type: Journal Article (International)

Journal: Acta Pharmaceutica Sciencia

Volume: 51

Year: 2009

Pages: 47-55

Metal Based Drugs: Current Use and Future Potential

Sanjay Kumar Bharti* and Sushil K. Singh

Publication Type: Journal Article (International)

Journal: Der Pharmacia Lettre

Volume: 1

Year: 2009

Pages: 39-51

Recent developments in the field of anticancer metallopharmaceuticals

Sanjay Kumar Bharti* and Sushil K. Singh,

Publication Type: Journal Article (International)

Journal: International Journal of PharmTech Research

Volume: 1

Year: 2009

Pages: 1406-1420

Antidepressant activity of ethanolic extract of Euphorbia thymifolia Linn. in the forced swimming test in rats

S. K. Singh*, T. Prabha, B. Kavitha, H. S. Chouhan and Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Pharmacologyonline

Volume: 2

Year: 2009

Pages: 967-970

Anti-inflammatory and Hepatoprotective activities of ethanolic extract of Euphorbia thymifolia Linn.

S. K. Singh*, T. Prabha, B. Kavitha, H. S. Chouhan and Sanjay Kumar Bharti

Publication Type: Journal Article (International)

Journal: Pharmacologyonline

Volume: 1

Year: 2009

Pages: 986-994

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